| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50014006 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_155157 |
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| Ki | 4408±n/a nM |
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| Citation |  Sunkel, CE; de Casa-Juana, MF; Santos, L; Gómez, MM; Villarroya, M; González-Morales, MA; Priego, JG; Ortega, MP 4-Alkyl-1,4-dihydropyridines derivatives as specific PAF-acether antagonists. J Med Chem33:3205-10 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50014006 |
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| n/a |
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| Name | BDBM50014006 |
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| Synonyms: | 2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-(2-methoxy-ethyl) ester 5-(2-methylsulfanyl-ethyl) ester | CHEMBL109083 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H25NO5S |
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| Mol. Mass. | 343.438 |
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| SMILES | COCCOC(=O)C1C(C)C(C(=O)OCCSC)=C(C)N=C1C |c:20,t:17| |
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| Structure | 
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