| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM82247 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_58990 |
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| Ki | 0.400000±n/a nM |
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| Citation |  Pettersson, I; Liljefors, T; Bøgesø, K Conformational analysis and structure-activity relationships of selective dopamine D-1 receptor agonists and antagonists of the benzazepine series. J Med Chem33:2197-204 (1990) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | D(1A) dopamine receptor | DOPAMINE D1 | DRD1_MOUSE | Dopamine D1 receptor | Dopamine receptor | Drd1 | Drd1a | Gpcr15 |
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| Type: | Enzyme |
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| Mol. Mass.: | 49613.93 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | Q61616 |
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| Residue: | 446 |
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| Sequence: | MAPNTSTMDETGLPVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNF
FVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDR
YWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLED
AEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKN
CQTTTGNGNPVECSQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGS
EETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIET
VSINNNGAVMFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKREEAGGIPKPLEKLSPAL
SVILDYDTDVSLEKIQPVTHSGQHST
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| BDBM82247 |
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| n/a |
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| Name | BDBM82247 |
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| Synonyms: | 8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol(SCH 23390) | CAS_87134-87-0 | CHEMBL2158641 | CHEMBL62 | SCH 23388 | SCH 23390 | SCH 23390 (R-enantiomer) | SCH 23390,R(+) |
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| Type | Small organic molecule |
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| Emp. Form. | C17H18ClNO |
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| Mol. Mass. | 287.784 |
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| SMILES | CN1CCc2cc(Cl)c(O)cc2[C@H](C1)c1ccccc1 |r| |
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| Structure | 
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