| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M1 |
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| Ligand | BDBM50010097 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_139068 |
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| Ki | 5.5±n/a nM |
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| Citation |  Hudkins, RL; DeHaven-Hudkins, DL; Stubbins, JF Muscarinic receptor binding profile of para-substituted caramiphen analogues. J Med Chem34:2984-9 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor M1 |
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| Name: | Muscarinic acetylcholine receptor M1 |
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| Synonyms: | ACM1_RAT | Cholinergic, muscarinic M1 | Chrm-1 | Chrm1 | cholinergic receptor, muscarinic 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51390.46 |
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| Organism: | RAT |
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| Description: | P08482 |
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| Residue: | 460 |
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| Sequence: | MNTSVPPAVSPNITVLAPGKGPWQVAFIGITTGLLSLATVTGNLLVLISFKVNTELKTVN
NYFLLSLACADLIIGTFSMNLYTTYLLMGHWALGTLACDLWLALDYVASNASVMNLLLIS
FDRYFSVTRPLSYRAKRTPRRAALMIGLAWLVSFVLWAPAILFWQYLVGERTVLAGQCYI
QFLSQPIITFGTAMAAFYLPVTVMCTLYWRIYRETENRARELAALQGSETPGKGGGSSSS
SERSQPGAEGSPESPPGRCCRCCRAPRLLQAYSWKEEEEEDEGSMESLTSSEGEEPGSEV
VIKMPMVDSEAQAPTKQPPKSSPNTVKRPTKKGRDRGGKGQKPRGKEQLAKRKTFSLVKE
KKAARTLSAILLAFILTWTPYNIMVLVSTFCKDCVPETLWELGYWLCYVNSTVNPMCYAL
CNKAFRDTFRLLLLCRWDKRRWRKIPKRPGSVHRTPSRQC
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| BDBM50010097 |
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| n/a |
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| Name | BDBM50010097 |
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| Synonyms: | 1-(4-Nitro-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester; hydrochloride | CHEMBL543382 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H26N2O4 |
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| Mol. Mass. | 334.41 |
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| SMILES | CCN(CC)CCOC(=O)C1(CCCC1)c1ccc(cc1)[N+]([O-])=O |
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| Structure | 
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