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TargetGag-Pol polyprotein [489-587]
LigandBDBM50368415
Substrate/Competitorn/a
Meas. Tech.ChEBML_157563
Ki 6.8±n/a nM
Citation Rich, DHPrasad, JVSun, CQGreen, JMueller, RHouseman, KMacKenzie, DMalkovsky, M New hydroxyethylamine HIV protease inhibitors that suppress viral replication. J Med Chem35:3803-12 (1992) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Gag-Pol polyprotein [489-587]
Name:Gag-Pol polyprotein [489-587]
Synonyms:Human immunodeficiency virus type 1 protease | POL_HV1H2 | Pol polyprotein | gag-pol
Type:Enzyme Subunit
Mol. Mass.:10781.16
Organism:Human immunodeficiency virus type 1
Description:P04585[489-587]
Residue:99
Sequence:
PQVTLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYD
QILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF
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  Blast E-value cutoff:
BDBM50368415
n/a
NameBDBM50368415
Synonyms:CHEMBL1790870 | CHEMBL3349481
TypeSmall organic molecule
Emp. Form.C51H71N7O10
Mol. Mass.942.1503
SMILES[H][C@@](O)(CN1CCCC1C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](C(C)C)C(=O)OC)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc1cccc(c1)-c1ccccc1)NC(=O)OC(C)(C)C
Structure
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