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TargetAdrenergic receptor beta
LigandBDBM50029050
Substrate/Competitorn/a
Meas. Tech.ChEBML_30208
Ki 720±n/a nM
Citation Chen GTKing MGusovsky FCreveling CRDaly JWChen BHNie JYKirk KL Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. J Med Chem 36:3947-55 (1994) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Adrenergic receptor beta
Name:Adrenergic receptor beta
Synonyms:Beta-2 adrenergic receptor
Type:PROTEIN
Mol. Mass.:46896.26
Organism:Rattus norvegicus
Description:ChEMBL_38603
Residue:418
Sequence:
MEPHGNDSDFLLAPNGSRAPGHDITQERDEAWVVGMAILMSVIVLAIVFGNVLVITAIAK
FERLQTVTNYFITSLACADLVMGLAVVPFGASHILMKMWNFGNFWCEFWTSIDVLCVTAS
IETLCVIAVDRYVAITSPFKYQSLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRATHKQ
AIDCYAKETCCDFFTNQAYAIASSIVSFYVPLVVMVFVYSRVFQVAKRQLQKIDKSEGRF
HAQNLSQVEQDGRSGHGLRSSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIRA
NLIPKEVYILLNWLGYVNSAFNPLIYCRSPDFRIAFQELLCLRRSSSKTYGNGYSSNSNG
RTDYTGEQSAYQLGQEKENELLCEEAPGMEGFVNCQGTVPSLSIDSQGRNCNTNDSPL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50029050
n/a
NameBDBM50029050
Synonyms:(-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((methylamino)methyl)benzyl alcohol | (-)-adrenaline | (R)-(-)-adrenaline | (R)-adrenaline | 4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol | Adrenalin | CHEMBL679 | EPINEPHRINE | adrenaline | levoepinephrine
TypeSmall organic molecule
Emp. Form.C9H13NO3
Mol. Mass.183.2044
SMILESCNC[C@H](O)c1ccc(O)c(O)c1 |r|
Structure
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