| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Plasminogen |
|---|
| Ligand | BDBM50286441 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_155050 (CHEMBL764369) |
|---|
| IC50 | 3700±n/a nM |
|---|
| Citation |  McConnell, RM; York, JL; Frizzell, D; Ezell, C Inhibition studies of some serine and thiol proteinases by new leupeptin analogues. J Med Chem36:1084-9 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Plasminogen |
|---|
| Name: | Plasminogen |
|---|
| Synonyms: | Activation peptide | PLG | PLMN_BOVIN | Plasmin heavy chain A | Plasmin heavy chain A, short form | Plasmin light chain B |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 91228.25 |
|---|
| Organism: | Bos taurus |
|---|
| Description: | ChEMBL_222778 |
|---|
| Residue: | 812 |
|---|
| Sequence: | MLPASPKMEHKAVVFLLLLFLKSGLGDLLDDYVNTQGASLLSLSRKNLAGRSVEDCAAKC
EEETDFVCRAFQYHSKEQQCVVMAENSKNTPVFRMRDVILYEKRIYLLECKTGNGQTYRG
TTAETKSGVTCQKWSATSPHVPKFSPEKFPLAGLEENYCRNPDNDENGPWCYTTDPDKRY
DYCDIPECEDKCMHCSGENYEGKIAKTMSGRDCQAWDSQSPHAHGYIPSKFPNKNLKMNY
CRNPDGEPRPWCFTTDPQKRWEFCDIPRCTTPPPSSGPKYQCLKGTGKNYGGTVAVTESG
HTCQRWSEQTPHKHNRTPENFPCKNLEENYCRNPNGEKAPWCYTTNSEVRWEYCTIPSCE
SSPLSTERMDVPVPPEQTPVPQDCYHGNGQSYRGTSSTTITGRKCQSWSSMTPHRHLKTP
ENYPNAGLTMNYCRNPDADKSPWCYTTDPRVRWEFCNLKKCSETPEQVPAAPQAPGVENP
PEADCMIGTGKSYRGKKATTVAGVPCQEWAAQEPHQHSIFTPETNPQSGLERNYCRNPDG
DVNGPWCYTMNPRKPFDYCDVPQCESSFDCGKPKVEPKKCSGRIVGGCVSKPHSWPWQVS
LRRSSRHFCGGTLISPKWVLTAAHCLDNILALSFYKVILGAHNEKVREQSVQEIPVSRLF
REPSQADIALLKLSRPAIITKEVIPACLPPPNYMVAARTECYITGWGETQGTFGEGLLKE
AHLPVIENKVCNRNEYLDGRVKPTELCAGHLIGGTDSCQGDSGGPLVCFEKDKYILQGVT
SWGLGCARPNKPGVYVRVSPYVPWIEETMRRN
|
|
|
|---|
| BDBM50286441 |
|---|
| n/a |
|---|
| Name | BDBM50286441 |
|---|
| Synonyms: | (S)-2-((S)-2-Acetylamino-4-(S)-methyl-pentanoylamino)-4-methyl-pentanoic acid (1-formyl-4-guanidino-butyl)-amide | (S)-2-Acetylamino-4-methyl-pentanoic acid [(R)-1-((S)-1-formyl-4-guanidino-butylcarbamoyl)-3-methyl-butyl]-amide | (S)-2-Acetylamino-4-methyl-pentanoic acid [(S)-1-((S)-1-formyl-4-guanidino-butylcarbamoyl)-3-methyl-butyl]-amide | (S)-2-[(S)-2-((S)-2-Acetylamino-4-methyl-pentanoylamino)-4-methyl-pentanoylamino]-5-guanidino-pentanoic acid | (S)-2-acetylamino-4-methyl-pentanoic acid [(S)-2-(1-formyl-4-guanidino-butylamino)-4-methyl-pentanoyl]-amide | 2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl-4-guanidino-butylcarbamoyl)-3-methyl-butyl]-amide | Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | CHEMBL129157 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H38N6O5 |
|---|
| Mol. Mass. | 442.5529 |
|---|
| SMILES | CC(C)C[C@H](NC(C)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
