| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50043720 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_136096 (CHEMBL745618) |
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| IC50 | 36±n/a nM |
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| Citation |  Bartosz-Bechowski, H; Davis, P; Zalewska, T; Slaninova, J; Porreca, F; Yamamura, HI; Hruby, VJ Cyclic enkephalin analogs with exceptional potency at peripheral delta opioid receptors. J Med Chem37:146-50 (1994) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50043720 |
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| n/a |
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| Name | BDBM50043720 |
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| Synonyms: | (S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(4-chloro-benzyl)-14,14-dimethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carbonyl]-amino}-3-phenyl-propionic acid | CHEMBL2372328 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H43ClN6O8S2 |
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| Mol. Mass. | 799.356 |
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| SMILES | CC1(C)SSC[C@H](NC(=O)[C@H](Cc2ccc(Cl)cc2)NC(=O)CNC(=O)[C@@H]1NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |
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| Structure | 
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