| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50453541 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_30471 (CHEMBL643132) |
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| Ki | 4.3±n/a nM |
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| Citation |  Gallo-Rodriguez, C; Ji, XD; Melman, N; Siegman, BD; Sanders, LH; Orlina, J; Fischer, B; Pu, Q; Olah, ME; van Galen, PJ Structure-activity relationships of N6-benzyladenosine-5'-uronamides as A3-selective adenosine agonists. J Med Chem37:636-46 (1994) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | AA3R_RAT | Adenosine A3 receptor | Adenosine receptor A2a and A3 | Adora3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36643.73 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_479910 |
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| Residue: | 320 |
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| Sequence: | MKANNTTTSALWLQITYITMEAAIGLCAVVGNMLVIWVVKLNRTLRTTTFYFIVSLALAD
IAVGVLVIPLAIAVSLEVQMHFYACLFMSCVLLVFTHASIMSLLAIAVDRYLRVKLTVRY
RTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKVTLELSQNSSTLSCHFRSVVGLDYMV
FFSFITWILIPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFL
FALCWLPLSIINFVSYFNVKIPEIAMCLGILLSHANSMMNPIVYACKIKKFKETYFVILR
ACRLCQTSDSLDSNLEQTTE
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|
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| BDBM50453541 |
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| n/a |
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| Name | BDBM50453541 |
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| Synonyms: | CHEMBL2113611 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H24N6O5 |
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| Mol. Mass. | 428.4418 |
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| SMILES | CCNC(=O)[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NCc3cccc(OC)c3)ncnc12 |r| |
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| Structure | 
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