Reaction Details | |||
---|---|---|---|
Report a problem with these data | |||
Target | Glutamyl aminopeptidase | ||
Ligand | BDBM50036820 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_32828 (CHEMBL646206) | ||
Ki | 1900±n/a nM | ||
Citation | Chauvel, EN; Coric, P; Llorens-Cortès, C; Wilk, S; Roques, BP; Fournié-Zaluski, MC Investigation of the active site of aminopeptidase A using a series of new thiol-containing inhibitors. J Med Chem37:1339-46 (1994) [PubMed] | ||
More Info.: | Get all data from this article, Assay Method | ||
Glutamyl aminopeptidase | |||
Name: | Glutamyl aminopeptidase | ||
Synonyms: | AMPE_HUMAN | AP-A | Aminopeptidase A | CD_antigen=CD249 | Differentiation antigen gp160 | EAP | ENPEP | Glutamyl aminopeptidase | ||
Type: | PROTEIN | ||
Mol. Mass.: | 109226.47 | ||
Organism: | Homo sapiens (Human) | ||
Description: | ChEMBL_32829 | ||
Residue: | 957 | ||
Sequence: |
| ||
BDBM50036820 | |||
n/a | |||
Name | BDBM50036820 | ||
Synonyms: | 2-(4-Carboxy-cyclohexyl)-1-mercaptomethyl-ethyl-ammonium | 4-(2-Amino-3-mercapto-propyl)-cyclohexanecarboxylic acid | CHEMBL26376 | ||
Type | Small organic molecule | ||
Emp. Form. | C10H19NO2S | ||
Mol. Mass. | 217.328 | ||
SMILES | NC(CS)CC1CCC(CC1)C(O)=O |(.78,-9.51,;.77,-7.97,;-.58,-7.2,;-1.91,-7.99,;2.1,-7.19,;3.43,-7.94,;3.43,-9.48,;4.76,-10.25,;6.11,-9.46,;6.1,-7.92,;4.75,-7.15,;7.42,-10.23,;7.42,-11.77,;8.77,-9.48,)| | ||
Structure |