| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50056629 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_145284 (CHEMBL751220) |
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| Ki | 210±n/a nM |
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| Citation |  Palmer, RB; Upthagrove, AL; Nelson, WL (E)- and (Z)-7-arylidenenaltrexones: synthesis and opioid receptor radioligand displacement assays. J Med Chem40:749-53 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50056629 |
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| n/a |
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| Name | BDBM50056629 |
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| Synonyms: | 4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-phenylphenyl)-(E)-methylidene]-(5R,13R,17S)-12-oxa-4-azapentacyclo[9.6.1.01,13.05,17.07,18]octadeca-7(18),8,10-trien-14-one | CHEMBL162048 | CHEMBL355188 |
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| Type | Small organic molecule |
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| Emp. Form. | C33H31NO4 |
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| Mol. Mass. | 505.6035 |
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| SMILES | Oc1ccc2C[C@H]3N(CC4CC4)CCC45[C@@H](Oc1c24)C(=O)C(C[C@@]35O)=Cc1ccc(cc1)-c1ccccc1 |w:25.31,THB:8:7:23:18.4.5| |
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| Structure | 
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