| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 1 |
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| Ligand | BDBM50062276 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_162504 (CHEMBL767332) |
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| IC50 | 1080±n/a nM |
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| Citation |  Camaioni, E; Boyer, JL; Mohanram, A; Harden, TK; Jacobson, KA Deoxyadenosine bisphosphate derivatives as potent antagonists at P2Y1 receptors. J Med Chem41:183-90 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 1 |
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| Name: | P2Y purinoceptor 1 |
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| Synonyms: | P2RY1 | P2RY1_MELGA |
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| Type: | n/a |
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| Mol. Mass.: | 41199.64 |
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| Organism: | Meleagris gallopavo |
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| Description: | n/a |
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| Residue: | 362 |
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| Sequence: | MTEALISAALNGTQPELLAGGWAAGNASTKCSLTKTGFQFYYLPTVYILVFITGFLGNSV
AIWMFVFHMRPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIF
HVNLYGSILFLTCISVHRYTGVVHPLKSLGRLKKKNAVYVSSLVWALVVAVIAPILFYSG
TGVRRNKTITCYDTTADEYLRSYFVYSMCTTVFMFCIPFIVILGCYGLIVKALIYKDLDN
SPLRRKSIYLVIIVLTVFAVSYLPFHVMKTLNLRARLDFQTPQMCAFNDKVYATYQVTRG
LASLNSCVDPILYFLAGDTFRRRLSRATRKSSRRSEPNVQSKSEEMTLNILTEYKQNGDT
SL
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| BDBM50062276 |
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| n/a |
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| Name | BDBM50062276 |
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| Synonyms: | CHEMBL55247 | Phosphoric acid mono-[5-(6-ethylamino-purin-9-yl)-2-phosphonooxymethyl-tetrahydro-furan-3-yl] ester |
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| Type | Small organic molecule |
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| Emp. Form. | C12H19N5O9P2 |
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| Mol. Mass. | 439.2549 |
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| SMILES | CCNc1ncnc2n(cnc12)C1CC(OP(O)(O)=O)C(COP(O)(O)=O)O1 |
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| Structure | 
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