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TargetMu-type opioid receptor
LigandBDBM50291970
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145302 (CHEMBL752837)
Ki 0.039000±n/a nM
Citation Thomas, JBFall, MJCooper, JBRothman, RBMascarella, SWXu, HPartilla, JSDersch, CMMcCullough, KBCantrell, BEZimmerman, DMCarroll, FI Identification of an opioid kappa receptor subtype-selective N-substituent for (+)-(3R,4R)-dimethyl-4-(3-hydroxyphenyl)piperidine. J Med Chem41:5188-97 (1999) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50291970
n/a
NameBDBM50291970
Synonyms:3-[(3S,4S)-3,4-Dimethyl-1-((E)-3-phenyl-allyl)-piperidin-4-yl]-phenol | CHEMBL150052
TypeSmall organic molecule
Emp. Form.C22H27NO
Mol. Mass.321.4559
SMILESC[C@@H]1CN(C\C=C\c2ccccc2)CC[C@]1(C)c1cccc(O)c1
Structure
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