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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Mu-type opioid receptor | ||
| Ligand | BDBM50001023 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_145274 (CHEMBL751210) | ||
| Ki | 0.100000±n/a nM | ||
| Citation |  Wentland, MP; Duan, W; Cohen, DJ; Bidlack, JM Selective protection and functionalization of morphine: synthesis and opioid receptor binding properties of 3-amino-3-desoxymorphine derivatives. J Med Chem43:3558-65 (2000) [PubMed] | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Mu-type opioid receptor | |||
| Name: | Mu-type opioid receptor | ||
| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 11165.58 | ||
| Organism: | GUINEA PIG | ||
| Description: | P97266 | ||
| Residue: | 98 | ||
| Sequence: |
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| BDBM50001023 | |||
| n/a | |||
| Name | BDBM50001023 | ||
| Synonyms: | (2R,6R,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | CHEMBL56585 | Cyclazocine | US10231963, Table B.9 | US10736890, Compound TABLE B.9 | US11534436, Compound Table B.9 | US9656961, Example 00126 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C18H25NO | ||
| Mol. Mass. | 271.3972 | ||
| SMILES | C[C@H]1[C@H]2Cc3ccc(O)cc3[C@]1(C)CCN2CC1CC1 |TLB:16:15:1:10.4.3| | ||
| Structure | 
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