| Reaction Details |
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 | Report a problem with these data |
| Target | Gamma-aminobutyric acid receptor subunit rho-1 |
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| Ligand | BDBM23183 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_68582 (CHEMBL679669) |
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| Kd | 2300±n/a nM |
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| Citation |  Chebib, M; Johnston, GA GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology. J Med Chem43:1427-47 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Gamma-aminobutyric acid receptor subunit rho-1 |
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| Name: | Gamma-aminobutyric acid receptor subunit rho-1 |
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| Synonyms: | GABA receptor rho-1 subunit | GABA-C receptor | GABRR1 | GBRR1_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 55892.34 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1456653 |
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| Residue: | 479 |
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| Sequence: | MLAVPNMRFGIFLLWWGWVLATESRMHWPGREVHEMSKKGRPQRQRREVHEDAHKQVSPI
LRRSPDITKSPLTKSEQLLRIDDHDFSMRPGFGGPAIPVGVDVQVESLDSISEVDMDFTM
TLYLRHYWKDERLSFPSTNNLSMTFDGRLVKKIWVPDMFFVHSKRSFIHDTTTDNVMLRV
QPDGKVLYSLRVTVTAMCNMDFSRFPLDTQTCSLEIESYAYTEDDLMLYWKKGNDSLKTD
ERISLSQFLIQEFHTTTKLAFYSSTGWYNRLYINFTLRRHIFFFLLQTYFPATLMVMLSW
VSFWIDRRAVPARVPLGITTVLTMSTIITGVNASMPRVSYIKAVDIYLWVSFVFVFLSVL
EYAAVNYLTTVQERKEQKLREKLPCTSGLPPPRTAMLDGNYSDGEVNDLDNYMPENGEKP
DRMMVQLTLASERSSPQRKSQRSSYVSMRIDTHAIDKYSRIIFPAAYILFNLIYWSIFS
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| BDBM23183 |
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| n/a |
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| Name | BDBM23183 |
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| Synonyms: | 5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL273481 | Muscimol | Pantherine |
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| Type | GABA Agonist |
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| Emp. Form. | C4H6N2O2 |
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| Mol. Mass. | 114.1026 |
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| SMILES | NCc1cc(=O)[nH]o1 |
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| Structure | 
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