| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 2-oxoglutarate receptor 1 |
|---|
| Ligand | BDBM50389799 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_151406 (CHEMBL754752) |
|---|
| Ki | 49±n/a nM |
|---|
| Citation |  Umino, T; Yoshioka, K; Saitoh, Y; Minakawa, N; Nakata, H; Matsuda, A Nucleosides and nucleotides. 200. Reinvestigation of 5'-N-ethylcarboxamidoadenosine derivatives: structure-activity relationships for P(3) purinoceptor-like proteins. J Med Chem44:208-14 (2001) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| 2-oxoglutarate receptor 1 |
|---|
| Name: | 2-oxoglutarate receptor 1 |
|---|
| Synonyms: | G protein-coupled receptor 80 | Gpr80 | OXGR1_RAT | Oxgr1 | P2y15 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 38385.93 |
|---|
| Organism: | Rattus norvegicus |
|---|
| Description: | ChEMBL_151406 |
|---|
| Residue: | 337 |
|---|
| Sequence: | MIETLDSPANDSDFLDYITALENCTDEQISFKMQYLPVIYSIIFLVGFPGNTVAISIYVF
KMRPWKSSTIIMLNLALTDLLYLTSLPFLIHYYASGENWIFGDFMCKFIRFGFHFNLYSS
ILFLTCFSLFRYIVIIHPMSCFSIQKTRWAVVACAGVWVISLVAVMPMTFLITSTTRTNR
SACLDLTSSDDLTTIKWYNLILTATTFCLPLLIVTLCYTTIISTLTHGPRTHSCFKQKAR
RLTILLLLVFYVCFLPFHILRVIRIESRLLSISCSIESHIHEAYIVSRPLAALNTFGNLL
LYVVVSNNFQQAFCSAVRCKAIGDLEQAKKDSCSNNP
|
|
|
|---|
| BDBM50389799 |
|---|
| n/a |
|---|
| Name | BDBM50389799 |
|---|
| Synonyms: | CHEMBL2070508 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H20N6O4 |
|---|
| Mol. Mass. | 348.3571 |
|---|
| SMILES | Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]([C@@H](O)[C@H]1O)C(=O)NC1CCCC1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
