Reaction Details | |||
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Target | Transient receptor potential cation channel subfamily V member 1 | ||
Ligand | BDBM50054471 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_215658 (CHEMBL821205) | ||
Ki | >5000±n/a nM | ||
Citation | López-Rodríguez, ML; Viso, A; Ortega-Gutiérrez, S; Lastres-Becker, I; González, S; Fernández-Ruiz, J; Ramos, JA Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors. J Med Chem44:4505-8 (2001) [PubMed] | ||
More Info.: | Get all data from this article, Assay Method | ||
Transient receptor potential cation channel subfamily V member 1 | |||
Name: | Transient receptor potential cation channel subfamily V member 1 | ||
Synonyms: | Capsaicin receptor | OTRPC1 | TRPV1_RAT | Transient receptor potential cation channel subfamily V member 1 (TRPV1) | Trpv1 | Vanilloid Receptor 1 (TRPV1, VR1) | Vanilloid VR1 | Vanilloid receptor | Vanilloid receptor 1 (VRI/TRPV1) | Vanilloid receptor type 1-like | Vanilloid receptor type 1-like (TrpV1/Vr1) | Vr1 | Vr1l | osm-9-like TRP channel 1 | ||
Type: | Transient Receptor | ||
Mol. Mass.: | 94956.12 | ||
Organism: | Rattus norvegicus (rat) | ||
Description: | O35433 | ||
Residue: | 838 | ||
Sequence: |
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BDBM50054471 | |||
n/a | |||
Name | BDBM50054471 | ||
Synonyms: | (5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy-phenyl)-amide | (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy-phenyl)-amide | (5Z,8Z,11Z,14Z)-N-(4-hydroxyphenyl)icosa-5,8,11,14-tetraenamide | (8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy-phenyl)-amide | AM-404 | AM404 | CHEMBL39878 | Icosa-5,8,11,14-tetraenoic acid (4-hydroxy-phenyl)-amide | N-(4-hydroxyphenyl)-(5Z,8Z,11Z,14Z)-icosatetra-5,8,11,14-enamide | N-(4-hydroxyphenyl)icosa-5,8,11,14-tetraenamide | cid_6604822 | ||
Type | Small organic molecule | ||
Emp. Form. | C26H37NO2 | ||
Mol. Mass. | 395.5775 | ||
SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)Nc1ccc(O)cc1 | ||
Structure |