| Reaction Details |
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 | Report a problem with these data |
| Target | P2X purinoceptor 5 |
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| Ligand | BDBM50118221 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147417 (CHEMBL750991) |
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| EC50 | >7000±n/a nM |
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| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2X purinoceptor 5 |
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| Name: | P2X purinoceptor 5 |
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| Synonyms: | ATP receptor | P2RX5_RAT | P2X5 | P2rx5 | Purinergic receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 51486.52 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_147417 |
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| Residue: | 455 |
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| Sequence: | MGQAAWKGFVLSLFDYKTAKFVVAKSKKVGLLYRVLQLIILLYLLIWVFLIKKSYQDIDT
SLQSAVVTKVKGVAYTNTTMLGERLWDVADFVIPSQGENVFFVVTNLIVTPNQRQGICAE
REGIPDGECSEDDDCHAGESVVAGHGLKTGRCLRVGNSTRGTCEIFAWCPVETKSMPTDP
LLKDAESFTISIKNFIRFPKFNFSKANVLETDNKHFLKTCHFSSTNLYCPIFRLGSIVRW
AGADFQDIALKGGVIGIYIEWDCDLDKAASKCNPHYYFNRLDNKHTHSISSGYNFRFARY
YRDPNGVEFRDLMKAYGIRFDVIVNGKAGKFSIIPTVINIGSGLALMGAGAFFCDLVLIY
LIRKSEFYRDKKFEKVRGQKEDANVEVEANEMEQERPEDEPLERVRQDEQSQELAQSGRK
QNSNCQVLLEPARFGLRENAIVNVKQSQILHPVKT
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| BDBM50118221 |
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| n/a |
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| Name | BDBM50118221 |
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| Synonyms: | 9H-purine derivative | CHEMBL132722 | DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER | alpha,beta-meATP |
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| Type | Small organic molecule |
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| Emp. Form. | C11H18N5O12P3 |
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| Mol. Mass. | 505.2082 |
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| SMILES | Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)CP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |
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| Structure | 
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