| Reaction Details |
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 | Report a problem with these data |
| Target | P2X purinoceptor 5 |
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| Ligand | BDBM50118219 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147416 (CHEMBL750990) |
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| EC50 | 40000±n/a nM |
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| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2X purinoceptor 5 |
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| Name: | P2X purinoceptor 5 |
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| Synonyms: | ATP receptor | P2RX5 | P2RX5_HUMAN | P2X5 | Purinergic receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47208.74 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_612725 |
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| Residue: | 422 |
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| Sequence: | MGQAGCKGLCLSLFDYKTEKYVIAKNKKVGLLYRLLQASILAYLVVWVFLIKKGYQDVDT
SLQSAVITKVKGVAFTNTSDLGQRIWDVADYVIPAQGENVFFVVTNLIVTPNQRQNVCAE
NEGIPDGACSKDSDCHAGEAVTAGNGVKTGRCLRRENLARGTCEIFAWCPLETSSRPEEP
FLKEAEDFTIFIKNHIRFPKFNFSKSNVMDVKDRSFLKSCHFGPKNHYCPIFRLGSVIRW
AGSDFQDIALEGGVIGINIEWNCDLDKAASECHPHYSFSRLDNKLSKSVSSGYNFRFARY
YRDAAGVEFRTLMKAYGIRFDVMVNGKGAFFCDLVLIYLIKKREFYRDKKYEEVRGLEDS
SQEAEDEASGLGLSEQLTSGPGLLGMPEQQELQEPPEAKRGSSSQKGNGSVCPQLLEPHR
ST
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| BDBM50118219 |
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| n/a |
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| Name | BDBM50118219 |
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| Synonyms: | Bz-ATP | CHEMBL339386 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H24N5O14P3 |
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| Mol. Mass. | 687.383 |
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| SMILES | Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1OC(=O)c1ccc(cc1)-c1ccccc1 |
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| Structure | 
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