| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 12 |
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| Ligand | BDBM50118232 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147742 (CHEMBL756289) |
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| EC50 | 1.1±n/a nM |
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| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 12 |
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| Name: | P2Y purinoceptor 12 |
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| Synonyms: | P2Y purinoceptor 12 | P2Y12_RAT | P2ry12 | P2y12 | Purinergic receptor P2Y12 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 39068.50 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_1454020 |
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| Residue: | 343 |
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| Sequence: | MEVPGANATSANTTSIPGTSTLCSRDYKITQVLFPLLYTVLFFAGLITNSLAMRIFFQIR
SKSNFIIFLKNTVISDLLMILTFPFKILSDAKLGAGHLRTLVCQVTSVTFYFTMYISISF
LGLITIDRYLKTTRPFKTSSPSNLLGAKILSVAIWAFMFLLSLPNMILTNRRPKDKDITK
CSFLKSEFGLVWHEIVNYICQVIFWINFLIVIVCYSLITKELYRSYVRTRGSAKAPKKRV
NIKVFIIIAVFFICFVPFHFARIPYTLSQTRAVFDCNAENTLFYVKESTLWLTSLNACLD
PFIYFFLCKSFRNSLMSMLRCSTSGANKKKGQEGGDPSEETPM
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| BDBM50118232 |
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| n/a |
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| Name | BDBM50118232 |
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| Synonyms: | 2-MeSATP | ATP, 2-meS | CHEMBL336208 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H18N5O13P3S |
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| Mol. Mass. | 553.273 |
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| SMILES | CSc1nc(N)c2ncn([C@@H]3O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]3O)c2n1 |
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| Structure | 
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