| Reaction Details |
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 | Report a problem with these data |
| Target | P2X purinoceptor 6 |
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| Ligand | BDBM85043 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147419 (CHEMBL750993) |
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| EC50 | >100000±n/a nM |
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| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2X purinoceptor 6 |
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| Name: | P2X purinoceptor 6 |
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| Synonyms: | ATP receptor | P2RX6_RAT | P2X6 | P2XM | P2rx6 | P2rxl1 | Purinergic receptor | Purinergic receptor P2X-like 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42451.11 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_147419 |
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| Residue: | 379 |
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| Sequence: | MASAVAAALVSWGFLDYKTEKYVMTRNCWVGISQRLLQLGVVVYVIGWALLAKKGYQEWD
MDPQISVITKLKGVSVTQVKELEKRLWDVADFVRPSQGENVFFLVTNFLVTPAQVQGRCP
EHPSVPLANCWADEDCPEGEMGTYSHGIKTGQCVAFNGTHRTCEIWSWCPVESSAVPRKP
LLAQAKNFTLFIKNTVTFNKFNFSRTNALDTWDNTYFKYCLYDSLSSPYCPVFRIGDLVA
MTGGDFEDLALLGGAVGINIHWDCNLDTKGSDCSPQYSFQLQERGYNFRTANYWWAASGV
ESRSLLKLYGIRFDILVTGQAGKFALIPTAITVGTGAAWLGMVTFLCDLLLLYVDREAGF
YWRTKYEEARAPKATTNSA
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| BDBM85043 |
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| n/a |
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| Name | BDBM85043 |
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| Synonyms: | CAS_149017-66-3 | CHEMBL69234 | NSC_6093163 | PPADS |
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| Type | Small organic molecule |
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| Emp. Form. | C14H14N3O12PS2 |
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| Mol. Mass. | 511.378 |
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| SMILES | Cc1nc(N=Nc2ccc(cc2S(O)(=O)=O)S(O)(=O)=O)c(COP(O)(O)=O)c(C=O)c1O |w:4.3| |
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| Structure | 
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