Reaction Details |
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Target | Corticotropin-releasing factor receptor 2 |
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Ligand | BDBM50119607 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_51272 (CHEMBL665763) |
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IC50 | 2.1±n/a nM |
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Citation | Rivier, J; Gulyas, J; Kirby, D; Low, W; Perrin, MH; Kunitake, K; DiGruccio, M; Vaughan, J; Reubi, JC; Waser, B; Koerber, SC; Martinez, V; Wang, L; Taché, Y; Vale, W Potent and long-acting corticotropin releasing factor (CRF) receptor 2 selective peptide competitive antagonists. J Med Chem45:4737-47 (2002) [PubMed] |
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More Info.: | Get all data from this article, Assay Method |
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Corticotropin-releasing factor receptor 2 |
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Name: | Corticotropin-releasing factor receptor 2 |
Synonyms: | CRF-R-2 | CRF-R2 | CRF2 Beta | CRFR-2 | CRFR2_RAT | CRH-R-2 | CRH-R2 | Corticotropin releasing factor receptor | Corticotropin-releasing factor receptor 2 | Corticotropin-releasing hormone receptor 2 | Crf2r | Crhr2 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 47697.09 |
Organism: | RAT |
Description: | CRF2 Beta 0 RAT::P47866 |
Residue: | 411 |
Sequence: | MDAALLLSLLEANCSLALAEELLLDGWGEPPDPEGPYSYCNTTLDQIGTCWPQSAPGALV
ERPCPEYFNGIKYNTTRNAYRECLENGTWASRVNYSHCEPILDDKQRKYDLHYRIALIIN
YLGHCVSVVALVAAFLLFLVLRSIRCLRNVIHWNLITTFILRNITWFLLQLIDHEVHEGN
EVWCRCVTTIFNYFVVTNFFWMFVEGCYLHTAIVMTYSTEHLRKWLFLFIGWCIPCPIIV
AWAVGKLYYENEQCWFGKEPGDLVDYIYQGPIILVLLINFVFLFNIVRILMTKLRASTTS
ETIQYRKAVKATLVLLPLLGITYMLFFVNPGEDDLSQIVFIYFNSFLQSFQGFFVSVFYC
FFNGEVRSALRKRWHRWQDHHALRVPVARAMSIPTSPTRISFHSIKQTAAV
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BDBM50119607 |
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n/a |
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Name | BDBM50119607 |
Synonyms: | CHEMBL440057 | E G P P I S I D L S L E L L R K M I E I E K Q E K E K Q Q A A N N R L L L D T I I-NH2(r/h CRF) | Human corticotropin releasing factor |
Type | Small organic molecule |
Emp. Form. | C208H343N59O64S2 |
Mol. Mass. | 4758.436 |
SMILES | n/a |
Structure |
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