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TargetMotilin receptor
LigandBDBM50344942
Substrate/Competitorn/a
Meas. Tech.ChEMBL_122661
EC50 400±n/a nM
Citation Li JJChao HGWang HTino JALawrence RMEwing WRMa ZYan MSlusarchyk DSeethala RSun HLi DBurford NTStoffel RHSalyan MELi CYWitkus MZhao NRich AGordon DA Discovery of a potent and novel motilin agonist. J Med Chem 47:1704-8 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Motilin receptor
Name:Motilin receptor
Synonyms:G-protein coupled receptor 38
Type:PROTEIN
Mol. Mass.:45365.95
Organism:Homo sapiens (Human)
Description:ChEMBL_122664
Residue:412
Sequence:
MGSPWNGSDGPEGAREPPWPALPPCDERRCSPFPLGALVPVTAVCLCLFVVGVSGNVVTV
MLIGRYRDMRTTTNLYLGSMAVSDLLILLGLPFDLYRLWRSRPWVFGPLLCRLSLYVGEG
CTYATLLHMTALSVERYLAICRPLRARVLVTRRRVRALIAVLWAVALLSAGPFLFLVGVE
QDPGISVVPGLNGTARIASSPLASSPPLWLSRAPPPSPPSGPETAEAAALFSRECRPSPA
QLGALRVMLWVTTAYFFLPFLCLSILYGLIGRELWSSRRPLRGPAASGRERGHRQTVRVL
LVVVLAFIICWLPFHVGRIIYINTEDSRMMYFSQYFNIVALQLFYLSASINPILYNLISK
KYRAAAFKLLLARKSRPRGFHRSRDTAGEVAGDTGGDTVGYTETSANVKTMG
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  Blast E-value cutoff:
BDBM50344942
n/a
NameBDBM50344942
Synonyms:CHEMBL532 | E-MYCIN E | ERYTHROMYCIN | ERYTHROMYCIN ETHYLSUCCINATE | Erycette | Erymax | Erythromycin A | Erythromycin C | Ilotycin | T-Stat
TypeSmall organic molecule
Emp. Form.C37H67NO13
Mol. Mass.733.9268
SMILESCC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O |r|
Structure
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