| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
|---|
| Ligand | BDBM50132714 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_305903 |
|---|
| IC50 | 304±n/a nM |
|---|
| Citation |  Lambert, DM; Fowler, CJ The endocannabinoid system: drug targets, lead compounds, and potential therapeutic applications. J Med Chem48:5059-87 (2005) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 1 |
|---|
| Name: | Cannabinoid receptor 1 |
|---|
| Synonyms: | Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_MOUSE | Cannabinoid CB1 receptor | Cannabinoid receptor | Cnr1 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 52842.52 |
|---|
| Organism: | Mus musculus (Mouse) |
|---|
| Description: | P47746 |
|---|
| Residue: | 473 |
|---|
| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEDNIQCGENFMDMECFMILNPSQQLAI
AVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHV
FHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCL
MWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILW
KAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPL
LAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTA
QPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
|
|
|
|---|
| BDBM50132714 |
|---|
| n/a |
|---|
| Name | BDBM50132714 |
|---|
| Synonyms: | (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenesulfonyl fluoride | CHEMBL112486 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H33FO2S |
|---|
| Mol. Mass. | 356.538 |
|---|
| SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCCS(F)(=O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
