| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50180044 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_329835 (CHEMBL854384) |
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| Ki | 70.8±n/a nM |
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| Citation |  Stern, E; Muccioli, GG; Millet, R; Goossens, JF; Farce, A; Chavatte, P; Poupaert, JH; Lambert, DM; Depreux, P; Hénichart, JP Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling. J Med Chem49:70-9 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50180044 |
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| n/a |
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| Name | BDBM50180044 |
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| Synonyms: | (RS)-N3-(1-phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide | CHEMBL426107 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H26N2O2 |
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| Mol. Mass. | 362.4647 |
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| SMILES | CCCCCn1cc(C(=O)NC(C)c2ccccc2)c(=O)c2ccccc12 |
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| Structure | 
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