| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Solute carrier family 15 member 1 |
|---|
| Ligand | BDBM50169199 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_363882 (CHEMBL863213) |
|---|
| IC50 | 810000±n/a nM |
|---|
| Citation |  Vig, BS; Stouch, TR; Timoszyk, JK; Quan, Y; Wall, DA; Smith, RL; Faria, TN Human PEPT1 pharmacophore distinguishes between dipeptide transport and binding. J Med Chem49:3636-44 (2006) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Solute carrier family 15 member 1 |
|---|
| Name: | Solute carrier family 15 member 1 |
|---|
| Synonyms: | Intestinal H(+)/peptide cotransporter | Oligopeptide transporter small intestine isoform | Oligopeptide transporter, small intestine isoform | PEPT1 | Peptide transporter 1 | S15A1_HUMAN | SLC15A1 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 78818.07 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1488839 |
|---|
| Residue: | 708 |
|---|
| Sequence: | MGMSKSHSFFGYPLSIFFIVVNEFCERFSYYGMRAILILYFTNFISWDDNLSTAIYHTFV
ALCYLTPILGALIADSWLGKFKTIVSLSIVYTIGQAVTSVSSINDLTDHNHDGTPDSLPV
HVVLSLIGLALIALGTGGIKPCVSAFGGDQFEEGQEKQRNRFFSIFYLAINAGSLLSTII
TPMLRVQQCGIHSKQACYPLAFGVPAALMAVALIVFVLGSGMYKKFKPQGNIMGKVAKCI
GFAIKNRFRHRSKAFPKREHWLDWAKEKYDERLISQIKMVTRVMFLYIPLPMFWALFDQQ
GSRWTLQATTMSGKIGALEIQPDQMQTVNAILIVIMVPIFDAVLYPLIAKCGFNFTSLKK
MAVGMVLASMAFVVAAIVQVEIDKTLPVFPKGNEVQIKVLNIGNNTMNISLPGEMVTLGP
MSQTNAFMTFDVNKLTRINISSPGSPVTAVTDDFKQGQRHTLLVWAPNHYQVVKDGLNQK
PEKGENGIRFVNTFNELITITMSGKVYANISSYNASTYQFFPSGIKGFTISSTEIPPQCQ
PNFNTFYLEFGSAYTYIVQRKNDSCPEVKVFEDISANTVNMALQIPQYFLLTCGEVVFSV
TGLEFSYSQAPSNMKSVLQAGWLLTVAVGNIIVLIVAGAGQFSKQWAEYILFAALLLVVC
VIFAIMARFYTYINPAEIEAQFDEDEKKNRLEKSNPYFMSGANSQKQM
|
|
|
|---|
| BDBM50169199 |
|---|
| n/a |
|---|
| Name | BDBM50169199 |
|---|
| Synonyms: | (S)-2-(2-Amino-acetylamino)-3-(3H-imidazol-4-yl)-propionic acid | 2-(2-Amino-acetylamino)-3-(3H-imidazol-4-yl)-propionic acid | CHEMBL93127 | Gly-His |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C8H12N4O3 |
|---|
| Mol. Mass. | 212.2059 |
|---|
| SMILES | NCC(=O)N[C@@H](Cc1cnc[nH]1)C(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
