| Reaction Details |
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 | Report a problem with these data |
| Target | Nociceptin receptor |
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| Ligand | BDBM50189257 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_378705 (CHEMBL853453) |
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| Ki | 0.300000±n/a nM |
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| Citation |  Crooks, PA; Kottayil, SG; Al-Ghananeem, AM; Byrn, SR; Butterfield, DA Opiate receptor binding properties of morphine-, dihydromorphine-, and codeine 6-O-sulfate ester congeners. Bioorg Med Chem Lett16:4291-5 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Nociceptin receptor |
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| Name: | Nociceptin receptor |
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| Synonyms: | OOR | OPRL1 | OPRX_CAVPO |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40796.89 |
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| Organism: | Cavia porcellus |
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| Description: | ChEMBL_444577 |
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| Residue: | 370 |
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| Sequence: | MESLFPAPFWEVLYGSHLQGNLSLLSPNHSGLPPHLLLNASHSAFLPLGLKVTIVGLYLA
VCIGGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQATDILLGFWPFGN
TLCKTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPIRALDVRTSSKAQAVNVAIWALALV
VGVPVAIMGSAQVEDEEIECLVEIPDPQDYWGPVFAVSIFLFSFIIPVLIISVCYSLMIR
RLHGVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLVQGLGVQPGSETTVAI
LRFCTALGYVNSCLNPILYAFLDENFKACFRKFCCASALHREMQVSDRVRSIAKDVALGC
KTTETVPRPA
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| BDBM50189257 |
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| n/a |
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| Name | BDBM50189257 |
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| Synonyms: | CHEMBL378753 | NalBzOH |
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| Type | Small organic molecule |
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| Emp. Form. | C26H27N3O4 |
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| Mol. Mass. | 445.5103 |
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| SMILES | Oc1ccc2CC3N(CC=C)CCC45[C@H](Oc1c24)C(CCC35O)=NNC(=O)c1ccccc1 |w:23.28,TLB:22:21:7.11.12:17.5.4,THB:8:7:21:17.5.4,16:17:21:7.11.12| |
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| Structure | 
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