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TargetProstaglandin E2 receptor EP1 subtype (EP1)
LigandBDBM50193931
Substrate/Competitorn/a
Meas. Tech.ChEMBL_424226
Ki>20000±n/a nM
Citation Belley MChan CCGareau YGallant MJuteau HHoude KLachance NLabelle MSawyer NTremblay NLamontagne SCarrière MCDenis DGreig GMSlipetz DGordon RChauret NLi CZamboni RJMetters KM Comparison between two classes of selective EP(3) antagonists and their biological activities. Bioorg Med Chem Lett 16:5639-42 (2006) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Prostaglandin E2 receptor EP1 subtype (EP1)
Name:Prostaglandin E2 receptor
Synonyms:PGE receptor, EP1 subtype | Prostaglandin E2 receptor EP1 subtype | Prostanoid EP1 receptor
Type:Enzyme
Mol. Mass.:41834.57
Organism:Homo sapiens (Human)
Description:P34995
Residue:402
Sequence:
MSPCGPLNLSLAGEATTCAAPWVPNTSAVPPSGASPALPIFSMTLGAVSNLLALALLAQA
AGRLRRRRSAATFLLFVASLLATDLAGHVIPGALVLRLYTAGRAPAGGACHFLGGCMVFF
GLCPLLLGCGMAVERCVGVTRPLLHAARVSVARARLALAAVAAVALAVALLPLARVGRYE
LQYPGTWCFIGLGPPGGWRQALLAGLFASLGLVALLAALVCNTLSGLALLRARWRRRSRR
PPPASGPDSRRRWGAHGPRSASASSASSIASASTFFGGSRSSGSARRARAHDVEMVGQLV
GIMVVSCICWSPMLVLVALAVGGWSSTSLQRPLFLAVRLASWNQILDPWVYILLRQAVLR
QLLRLLPPRAGAKGGPAGLGLTPSAWEASSLRSSRHSGLSHF
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  Blast E-value cutoff:
BDBM50193931
n/a
NameBDBM50193931
Synonyms:3-(2-(4-(benzyloxy)-3-methoxycinnamyl)phenyl)acrylic acid | CHEMBL218626
TypeSmall organic molecule
Emp. Form.C26H24O4
Mol. Mass.400.4664
SMILESCOc1cc(\C=C\Cc2ccccc2\C=C\C(O)=O)ccc1OCc1ccccc1
Structure
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