| Reaction Details |
|---|
 | Report a problem with these data |
| Target | MO15-related protein kinase Pfmrk |
|---|
| Ligand | BDBM15203 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_456708 (CHEMBL923066) |
|---|
| IC50 | >500000±n/a nM |
|---|
| Citation |  Woodard, CL; Keenan, SM; Gerena, L; Welsh, WJ; Geyer, JA; Waters, NC Evaluation of broad spectrum protein kinase inhibitors to probe the architecture of the malarial cyclin dependent protein kinase Pfmrk. Bioorg Med Chem Lett17:4961-6 (2007) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| MO15-related protein kinase Pfmrk |
|---|
| Name: | MO15-related protein kinase Pfmrk |
|---|
| Synonyms: | Protein kinase Pfmrk |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 37992.30 |
|---|
| Organism: | Plasmodium falciparum |
|---|
| Description: | ChEMBL_640752 |
|---|
| Residue: | 324 |
|---|
| Sequence: | MENNSTERYIFKPNFLGEGSYGKVYKAYDTILKKEVAIKKMKLNEISNYIDDCGINFVLL
REIKIMKEIKHKNIMSALDLYCEKDYINLVMEIMDYDLSKIINRKIFLTDSQKKCILLQI
LNGLNVLHKYYFMHRDLSPANIFINKKGEVKLADFGLCTKYGYDMYSDKLFRDKYKKNLN
LTSKVVTLWYRAPELLLGSNKYNSSIDMWSFGCIFAELLLQKALFPGENEIDQLGKIFFL
LGTPNENNWPEALCLPLYTEFTKATKKDFKTYFKIDDDDCIDLLTSFLKLNAHERISAED
AMKHRYFFNDPLPCDISQLPFNDL
|
|
|
|---|
| BDBM15203 |
|---|
| n/a |
|---|
| Name | BDBM15203 |
|---|
| Synonyms: | 5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL75773 | Isoquinoline-5-sulfonic acid piperazin-1 ylamide | isoquinoline-5-sulfonamide 18 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C13H15N3O2S |
|---|
| Mol. Mass. | 277.342 |
|---|
| SMILES | O=S(=O)(N1CCNCC1)c1cccc2cnccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
