| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Purinergic receptor P2Y2 |
|---|
| Ligand | BDBM50336791 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_463988 |
|---|
| IC50 | 14000±n/a nM |
|---|
| Citation |  Weyler S; Baqi Y; Hillmann P; Kaulich M; Hunder AM; Müller IA; Müller CE Combinatorial synthesis of anilinoanthraquinone derivatives and evaluation as non-nucleotide-derived P2Y2 receptor antagonists. Bioorg Med Chem Lett 18:223-7 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Purinergic receptor P2Y2 |
|---|
| Name: | Purinergic receptor P2Y2 |
|---|
| Synonyms: | ATP receptor | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | Purinergic receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 42202.78 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | ChEMBL_587770 |
|---|
| Residue: | 373 |
|---|
| Sequence: | MAADLEPWNSTINGTWEGDELGYKCRFNEDFKYVLLPVSYGVVCVLGLCLNVVALYIFLC
RLKTWNASTTYMFHLAVSDSLYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCS
ILFLTCISVHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTR
ITCHDTSARELFSHFVAYSSVMLGLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAK
RKSVRTIALVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPLASANSC
LDPVLYFLAGQRLVRFARDAKPPTEPTPSPQARRKLGLHRPNRTVRKDLSVSSDDSRRTE
STPAGSETKDIRL
|
|
|
|---|
| BDBM50336791 |
|---|
| n/a |
|---|
| Name | BDBM50336791 |
|---|
| Synonyms: | CHEMBL402239 | sodium 1-amino-4-(2,3-dimethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C22H17N2O5S |
|---|
| Mol. Mass. | 421.446 |
|---|
| SMILES | Cc1cccc(Nc2cc(c(N)c3C(=O)c4ccccc4C(=O)c23)S([O-])(=O)=O)c1C |
|---|
| Structure | 
|
|---|
Search and Browse
