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TargetP2Y purinoceptor 4
LigandBDBM50336767
Substrate/Competitorn/a
Meas. Tech.ChEMBL_463992 (CHEMBL929979)
IC50 50000±n/a nM
Citation Weyler, SBaqi, YHillmann, PKaulich, MHunder, AMMüller, IAMüller, CE Combinatorial synthesis of anilinoanthraquinone derivatives and evaluation as non-nucleotide-derived P2Y2 receptor antagonists. Bioorg Med Chem Lett18:223-7 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
P2Y purinoceptor 4
Name:P2Y purinoceptor 4
Synonyms:NRU | P2P | P2RY4 | P2RY4_HUMAN | P2Y purinoceptor 4 | P2Y4 | Pyrimidinergic receptor P2Y4 | UNR | Uridine nucleotide receptor
Type:PROTEIN
Mol. Mass.:40977.17
Organism:Homo sapiens (Human)
Description:ChEMBL_751027
Residue:365
Sequence:
MASTESSLLRSLGLSPGPGSSEVELDCWFDEDFKFILLPVSYAVVFVLGLGLNAPTLWLF
IFRLRPWDATATYMFHLALSDTLYVLSLPTLIYYYAAHNHWPFGTEICKFVRFLFYWNLY
CSVLFLTCISVHRYLGICHPLRALRWGRPRLAGLLCLAVWLVVAGCLVPNLFFVTTSNKG
TTVLCHDTTRPEEFDHYVHFSSAVMGLLFGVPCLVTLVCYGLMARRLYQPLPGSAQSSSR
LRSLRTIAVVLTVFAVCFVPFHITRTIYYLARLLEADCRVLNIVNVVYKVTRPLASANSC
LDPVLYLLTGDKYRRQLRQLCGGGKPQPRTAASSLALVSLPEDSSCRWAATPQDSSCSTP
RADRL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50336767
n/a
NameBDBM50336767
Synonyms:CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
TypeSmall organic molecule
Emp. Form.C21H15N2O6S
Mol. Mass.423.419
SMILESCOc1ccccc1Nc1cc(c(N)c2C(=O)c3ccccc3C(=O)c12)S([O-])(=O)=O
Structure
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