| Reaction Details |
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 | Report a problem with these data |
| Target | Transcriptional activator protein LuxR |
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| Ligand | BDBM50373052 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_466368 (CHEMBL932480) |
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| IC50 | 6400±n/a nM |
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| Citation |  Frezza, M; Soulère, L; Reverchon, S; Guiliani, N; Jerez, C; Queneau, Y; Doutheau, A Synthetic homoserine lactone-derived sulfonylureas as inhibitors of Vibrio fischeri quorum sensing regulator. Bioorg Med Chem16:3550-6 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Transcriptional activator protein LuxR |
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| Name: | Transcriptional activator protein LuxR |
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| Synonyms: | LUXR_ALIFS | luxR |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28563.86 |
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| Organism: | Vibrio fischeri |
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| Description: | ChEMBL_831639 |
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| Residue: | 250 |
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| Sequence: | MKNINADDTYRIINKIKACRSNNDINQCLSDMTKMVHCEYYLLAIIYPHSMVKSDISILD
NYPKKWRQYYDDANLIKYDPIVDYSNSNHSPINWNIFENNAVNKKSPNVIKEAKTSGLIT
GFSFPIHTANNGFGMLSFAHSEKDNYIDSLFLHACMNIPLIVPSLVDNYRKINIANNKSN
NDLTKREKECLAWACEGKSSWDISKILGCSERTVTFHLTNAQMKLNTTNRCQSISKAILT
GAIDCPYFKN
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| BDBM50373052 |
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| n/a |
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| Name | BDBM50373052 |
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| Synonyms: | CHEMBL404926 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H14N2O4S |
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| Mol. Mass. | 270.305 |
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| SMILES | O=C1OCCC1NS(=O)(=O)NCc1ccccc1 |w:5.6| |
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| Structure | 
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