Reaction Details | |||
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Target | Cyclin-dependent kinase 5 activator 1 | ||
Ligand | BDBM50005298 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_473638 (CHEMBL937655) | ||
IC50 | 20±n/a nM | ||
Citation | Fedorov, O; Marsden, B; Pogacic, V; Rellos, P; Müller, S; Bullock, AN; Schwaller, J; Sundström, M; Knapp, S A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases. Proc Natl Acad Sci U S A104:20523-8 (2007) [PubMed] Article | ||
More Info.: | Get all data from this article, Assay Method | ||
Cyclin-dependent kinase 5 activator 1 | |||
Name: | Cyclin-dependent kinase 5 activator 1 | ||
Synonyms: | CD5R1_HUMAN | CDK5R | CDK5R1 | Cyclin-Dependent Kinase 5 Activator 1, p35 | Cyclin-dependent kinase 5 (CDK5/p25) | Cyclin-dependent kinase 5 regulatory subunit 1 | NCK5A | TPKII regulatory subunit | p35 | ||
Type: | Enzyme Subunit | ||
Mol. Mass.: | 34077.43 | ||
Organism: | Homo sapiens (Human) | ||
Description: | Q15078 | ||
Residue: | 307 | ||
Sequence: |
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BDBM50005298 | |||
n/a | |||
Name | BDBM50005298 | ||
Synonyms: | CHEMBL337300 | ||
Type | Small organic molecule | ||
Emp. Form. | C16H10IN3O2 | ||
Mol. Mass. | 403.174 | ||
SMILES | Oc1[nH]c2ccc(I)cc2c1-c1[nH]c2ccccc2c1N=O |(3.16,-9.8,;3.62,-8.34,;5.09,-7.85,;5.07,-6.31,;6.21,-5.28,;5.89,-3.79,;4.42,-3.31,;4.09,-1.8,;3.27,-4.35,;3.6,-5.84,;2.71,-7.09,;1.17,-7.1,;.26,-8.36,;-1.21,-7.89,;-2.54,-8.66,;-3.87,-7.89,;-3.87,-6.35,;-2.54,-5.58,;-1.21,-6.35,;.26,-5.86,;.73,-4.39,;-.32,-3.25,)| | ||
Structure |