| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50377702 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_479928 (CHEMBL929251) |
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| Ki | 19±n/a nM |
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| Citation |  Worm, K; Zhou, QJ; Saeui, CT; Green, RC; Cassel, JA; Stabley, GJ; DeHaven, RN; Conway-James, N; LaBuda, CJ; Koblish, M; Little, PJ; Dolle, RE Sulfamoyl benzamides as novel CB2 cannabinoid receptor ligands. Bioorg Med Chem Lett18:2830-5 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50377702 |
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| n/a |
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| Name | BDBM50377702 |
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| Synonyms: | CHEMBL258244 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H30N2O4S |
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| Mol. Mass. | 418.55 |
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| SMILES | Cc1ccc(cc1S(=O)(=O)N1CCOCC1)C(=O)NC12CC3CC(CC(C3)C1)C2 |TLB:22:23:27:20.21.26,26:21:28:27.25.24,26:25:28:20.21.22,THB:22:21:27:28.23.24| |
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| Structure | 
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