| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50260710 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_552264 (CHEMBL995594) |
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| Ki | 242±n/a nM |
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| Citation |  Omura, H; Kawai, M; Shima, A; Iwata, Y; Ito, F; Masuda, T; Ohta, A; Makita, N; Omoto, K; Sugimoto, H; Kikuchi, A; Iwata, H; Ando, K The SAR studies of novel CB2 selective agonists, benzimidazolone derivatives. Bioorg Med Chem Lett18:3310-4 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50260710 |
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| n/a |
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| Name | BDBM50260710 |
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| Synonyms: | (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-2-oxo-3-(2-(pyrrolidin-1-yl)ethyl)-2,3-dihydrobenzo[d]imidazole-1-carboxamide | CHEMBL524818 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H29N5O3 |
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| Mol. Mass. | 387.476 |
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| SMILES | CC(C)(C)[C@H](NC(=O)n1c2ccccc2n(CCN2CCCC2)c1=O)C(N)=O |r| |
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| Structure | 
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