| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
|---|
| Ligand | BDBM50260753 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_552265 (CHEMBL995595) |
|---|
| EC50 | 2±n/a nM |
|---|
| Citation |  Omura, H; Kawai, M; Shima, A; Iwata, Y; Ito, F; Masuda, T; Ohta, A; Makita, N; Omoto, K; Sugimoto, H; Kikuchi, A; Iwata, H; Ando, K The SAR studies of novel CB2 selective agonists, benzimidazolone derivatives. Bioorg Med Chem Lett18:3310-4 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 2 |
|---|
| Name: | Cannabinoid receptor 2 |
|---|
| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 39690.94 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P34972 |
|---|
| Residue: | 360 |
|---|
| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
|
|
|
|---|
| BDBM50260753 |
|---|
| n/a |
|---|
| Name | BDBM50260753 |
|---|
| Synonyms: | (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(3-hydroxy-3-methylbutyl)-2-oxo-2,3-dihydrobenzo[d]imidazole-1-carboxamide | CHEMBL506652 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H28N4O4 |
|---|
| Mol. Mass. | 376.45 |
|---|
| SMILES | CC(C)(O)CCn1c2ccccc2n(C(=O)N[C@H](C(N)=O)C(C)(C)C)c1=O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
