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TargetFatty acid-binding protein, liver
LigandBDBM50292627
Substrate/Competitorn/a
Meas. Tech.ChEMBL_555395 (CHEMBL964792)
Ki 12900±n/a nM
Citation Chuang, SVelkov, THorne, JPorter, CJScanlon, MJ Characterization of the drug binding specificity of rat liver fatty acid binding protein. J Med Chem51:3755-64 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, liver
Name:Fatty acid-binding protein, liver
Synonyms:FABPL_RAT | Fabp1 | Fatty acid-binding protein, liver | Liver fatty acid binding protein (rat L-FABP)
Type:Protein
Mol. Mass.:14274.39
Organism:Rattus norvegicus (Rat)
Description:rat L-FABP
Residue:127
Sequence:
MNFSGKYQVQSQENFEPFMKAMGLPEDLIQKGKDIKGVSEIVHEGKKVKLTITYGSKVIH
NEFTLGEECELETMTGEKVKAVVKMEGDNKMVTTFKGIKSVTEFNGDTITNTMTLGDIVY
KRVSKRI
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BDBM50292627
n/a
NameBDBM50292627
Synonyms:(RS)-9-chloro-6-(2-chlorophenyl)-4-hydroxy-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen-3-one | 7-Chloro-5-(2-chloro-phenyl)-3-hydroxy-1,3-dihydro-benzo[e][1,4]diazepin-2-one | 7-Chloro-5-(2-chloro-phenyl)-3-hydroxy-1,3-dihydro-benzo[e][1,4]diazepin-2-one (lorazepam) | 7-chloro-5-(2-chlorophenyl)-3-hydroxy-1H-benzo[e][1,4]diazepin-2(3H)-one | Ativan | CHEMBL580 | LORAZEPAM | LORAZEPAM7-Chloro-5-(2-chloro-phenyl)-3-hydroxy-1,3-dihydro-benzo[e][1,4]diazepin-2-one | Loraz | Lorazepam intensol | Lorazepam preservative free | WY-4036
TypeSmall organic molecule
Emp. Form.C15H10Cl2N2O2
Mol. Mass.321.158
SMILESOC1N=C(c2ccccc2Cl)c2cc(Cl)ccc2NC1=O |t:2|
Structure
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