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TargetCannabinoid receptor 2
LigandBDBM50265757
Substrate/Competitorn/a
Meas. Tech.ChEMBL_560595
Ki 342±n/a nM
Citation Markt PFeldmann CRollinger JMRaduner SSchuster DKirchmair JDistinto SSpitzer GMWolber GLaggner CAltmann KHLanger TGertsch J Discovery of novel CB2 receptor ligands by a pharmacophore-based virtual screening workflow. J Med Chem 52:369-78 (2009) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:39690.94
Organism:Homo sapiens (Human)
Description:P34972
Residue:360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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BDBM50265757
n/a
NameBDBM50265757
Synonyms:4-(2,6-dimethoxy-4-(2-methyloctan-2-yl)phenyl)tetrahydro-2H-pyran-4-ol | CHEMBL495546
TypeSmall organic molecule
Emp. Form.C22H36O4
Mol. Mass.364.5188
SMILESCCCCCCC(C)(C)c1cc(OC)c(c(OC)c1)C1(O)CCOCC1
Structure
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