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TargetMu-type opioid receptor
LigandBDBM50248990
Substrate/Competitorn/a
Meas. Tech.ChEMBL_543319
Ki 3.3±n/a nM
Citation Moynihan HJales ARGreedy BMRennison DBroadbear JHPurington LTraynor JRWoods JHLewis JWHusbands SM 14 beta-O-cinnamoylnaltrexone and related dihydrocodeinones are mu opioid receptor partial agonists with predominant antagonist activity. J Med Chem 52:1553-7 (2009) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50248990
n/a
NameBDBM50248990
Synonyms:14beta-(4-Methylcinnamoyloxy)-N-cyclopropylmethyl-7,8-dihydronormorphinone | CHEMBL474641
TypeSmall organic molecule
Emp. Form.C30H31NO5
Mol. Mass.485.5708
SMILESCc1ccc(\C=C\C(=O)O[C@]23CCC(=O)[C@@H]4Oc5c6c(C[C@H]2N(CC2CC2)CC[C@@]346)ccc5O)cc1 |r|
Structure
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