| Reaction Details |
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 | Report a problem with these data |
| Target | Galectin-8 |
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| Ligand | BDBM50326596 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_661837 (CHEMBL1252153) |
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| Kd | 66000±n/a nM |
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| Citation |  Salameh, BA; Cumpstey, I; Sundin, A; Leffler, H; Nilsson, UJ 1H-1,2,3-triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors. Bioorg Med Chem18:5367-78 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Galectin-8 |
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| Name: | Galectin-8 |
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| Synonyms: | Gal-8 | LEG8_HUMAN | LGALS8 | PCTA-1 | Po66 carbohydrate-binding protein | Po66-CBP | Prostate carcinoma tumor antigen 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 35814.23 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1454625 |
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| Residue: | 317 |
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| Sequence: | MMLSLNNLQNIIYNPVIPFVGTIPDQLDPGTLIVIRGHVPSDADRFQVDLQNGSSMKPRA
DVAFHFNPRFKRAGCIVCNTLINEKWGREEITYDTPFKREKSFEIVIMVLKDKFQVAVNG
KHTLLYGHRIGPEKIDTLGIYGKVNIHSIGFSFSSDLQSTQASSLELTEISRENVPKSGT
PQLRLPFAARLNTPMGPGRTVVVKGEVNANAKSFNVDLLAGKSKDIALHLNPRLNIKAFV
RNSFLQESWGEEERNITSFPFSPGMYFEMIIYCDVREFKVAVNGVHSLEYKHRFKELSSI
DTLEINGDIHLLEVRSW
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| BDBM50326596 |
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| n/a |
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| Name | BDBM50326596 |
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| Synonyms: | CHEMBL1253187 | Di-(3-deoxy-3-(4-((allylamino)carbonyl)-1H-1,2,3-triazol-1-yl)-beta-D-galactopyranosyl)sulfane |
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| Type | Small organic molecule |
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| Emp. Form. | C24H34N8O10S |
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| Mol. Mass. | 626.639 |
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| SMILES | OC[C@H]1O[C@@H](S[C@@H]2O[C@H](CO)[C@H](O)[C@@H]([C@H]2O)n2cc(nn2)C(=O)NCC=C)[C@H](O)[C@H]([C@H]1O)n1cc(nn1)C(=O)NCC=C |r| |
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| Structure | 
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