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TargetMotilin receptor
LigandBDBM50344942
Substrate/Competitorn/a
Meas. Tech.ChEMBL_664665
EC50 1200±n/a nM
Citation Liu YLi YChen YZheng HClaypool MMyles DCCarreras CW 9-Dihydroerythromycins as non-antibiotic motilin receptor agonists. Bioorg Med Chem Lett 20:5658-61 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Motilin receptor
Name:Motilin receptor
Synonyms:n/a
Type:n/a
Mol. Mass.:43771.25
Organism:Oryctolagus cuniculus
Description:n/a
Residue:400
Sequence:
MGSPWNGSDGPEDAREPPWAALPPCDERRCSPFPLGTLVPVTAVCLGLFAVGVSGNVVTV
LLIGRYRDMRTTTNLYLGSMAVSDLLILLGLPFDLYRLWRSRPWVFGQLLCRLSLYVGEG
CTYASLLHMTALSVERYLAICRPLRARVLVTRRRVRALIAALWAVALLSAGPFFFLVGVE
QDPAVFAAPDRNGTVPLDPSSPAPASPPSGPGAEAAALFSRECRPSRAQLGLLRVMLWVT
TAYFFLPFLCLSILYGLIARQLWRGRGPLRGPAATGRERGHRQTVRVLLVVVLAFIVCWL
PFHVGRIIYINTQDSRMMYFSQYFNIVALQLFYLSASINPILYNLISKKYRAAARRLLRE
SRAGPSGVCGSRGPEQDVAGDTGGDTAGCTETSANTKTAA
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  Blast E-value cutoff:
BDBM50344942
n/a
NameBDBM50344942
Synonyms:CHEMBL532 | E-MYCIN E | ERYTHROMYCIN | ERYTHROMYCIN ETHYLSUCCINATE | Erycette | Erymax | Erythromycin A | Erythromycin C | Ilotycin | T-Stat
TypeSmall organic molecule
Emp. Form.C37H67NO13
Mol. Mass.733.9268
SMILESCC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O |r|
Structure
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