| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 4 |
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| Ligand | BDBM50227020 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_718669 (CHEMBL1680820) |
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| IC50 | 21800±n/a nM |
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| Citation |  Baqi, Y; Hausmann, R; Rosefort, C; Rettinger, J; Schmalzing, G; Müller, CE Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem54:817-30 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 4 |
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| Name: | P2Y purinoceptor 4 |
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| Synonyms: | NRU | P2P | P2RY4 | P2RY4_HUMAN | P2Y purinoceptor 4 | P2Y4 | Pyrimidinergic receptor P2Y4 | UNR | Uridine nucleotide receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40977.17 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_751027 |
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| Residue: | 365 |
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| Sequence: | MASTESSLLRSLGLSPGPGSSEVELDCWFDEDFKFILLPVSYAVVFVLGLGLNAPTLWLF
IFRLRPWDATATYMFHLALSDTLYVLSLPTLIYYYAAHNHWPFGTEICKFVRFLFYWNLY
CSVLFLTCISVHRYLGICHPLRALRWGRPRLAGLLCLAVWLVVAGCLVPNLFFVTTSNKG
TTVLCHDTTRPEEFDHYVHFSSAVMGLLFGVPCLVTLVCYGLMARRLYQPLPGSAQSSSR
LRSLRTIAVVLTVFAVCFVPFHITRTIYYLARLLEADCRVLNIVNVVYKVTRPLASANSC
LDPVLYLLTGDKYRRQLRQLCGGGKPQPRTAASSLALVSLPEDSSCRWAATPQDSSCSTP
RADRL
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| BDBM50227020 |
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| n/a |
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| Name | BDBM50227020 |
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| Synonyms: | CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate |
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| Type | Small organic molecule |
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| Emp. Form. | C20H12ClN2O5S |
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| Mol. Mass. | 427.838 |
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| SMILES | Nc1c(cc(Nc2cccc(Cl)c2)c2C(=O)c3ccccc3C(=O)c12)S([O-])(=O)=O |
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| Structure | 
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