| Reaction Details |
|---|
 | Report a problem with these data |
| Target | P2Y purinoceptor 6 |
|---|
| Ligand | BDBM50268725 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_718670 (CHEMBL1680821) |
|---|
| IC50 | 5300±n/a nM |
|---|
| Citation |  Baqi, Y; Hausmann, R; Rosefort, C; Rettinger, J; Schmalzing, G; Müller, CE Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem54:817-30 (2012) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| P2Y purinoceptor 6 |
|---|
| Name: | P2Y purinoceptor 6 |
|---|
| Synonyms: | P2RY6 | P2RY6_HUMAN | P2Y purinoceptor 6 | P2Y6 | Pyrimidinergic receptor P2Y6 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 36452.29 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1511151 |
|---|
| Residue: | 328 |
|---|
| Sequence: | MEWDNGTGQALGLPPTTCVYRENFKQLLLPPVYSAVLAAGLPLNICVITQICTSRRALTR
TAVYTLNLALADLLYACSLPLLIYNYAQGDHWPFGDFACRLVRFLFYANLHGSILFLTCI
SFQRYLGICHPLAPWHKRGGRRAAWLVCVAVWLAVTTQCLPTAIFAATGIQRNRTVCYDL
SPPALATHYMPYGMALTVIGFLLPFAALLACYCLLACRLCRQDGPAEPVAQERRGKAARM
AVVVAAAFAISFLPFHITKTAYLAVRSTPGVPCTVLEAFAAAYKGTRPFASANSVLDPIL
FYFTQKKFRRRPHELLQKLTAKWQRQGR
|
|
|
|---|
| BDBM50268725 |
|---|
| n/a |
|---|
| Name | BDBM50268725 |
|---|
| Synonyms: | CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H13N2O6S |
|---|
| Mol. Mass. | 409.393 |
|---|
| SMILES | Nc1c(cc(Nc2ccc(O)cc2)c2C(=O)c3ccccc3C(=O)c12)S([O-])(=O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
