| Reaction Details |
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 | Report a problem with these data |
| Target | Pyrimidinergic receptor P2Y6 |
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| Ligand | BDBM50227020 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_718670 |
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| IC50 | >10000±n/a nM |
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| Citation |  Baqi Y; Hausmann R; Rosefort C; Rettinger J; Schmalzing G; Müller CE Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem 54:817-30 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Pyrimidinergic receptor P2Y6 |
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| Name: | Pyrimidinergic receptor P2Y6 |
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| Synonyms: | P2Y purinoceptor 6 | P2Y6 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36452.29 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1511151 |
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| Residue: | 328 |
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| Sequence: | MEWDNGTGQALGLPPTTCVYRENFKQLLLPPVYSAVLAAGLPLNICVITQICTSRRALTR
TAVYTLNLALADLLYACSLPLLIYNYAQGDHWPFGDFACRLVRFLFYANLHGSILFLTCI
SFQRYLGICHPLAPWHKRGGRRAAWLVCVAVWLAVTTQCLPTAIFAATGIQRNRTVCYDL
SPPALATHYMPYGMALTVIGFLLPFAALLACYCLLACRLCRQDGPAEPVAQERRGKAARM
AVVVAAAFAISFLPFHITKTAYLAVRSTPGVPCTVLEAFAAAYKGTRPFASANSVLDPIL
FYFTQKKFRRRPHELLQKLTAKWQRQGR
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| BDBM50227020 |
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| n/a |
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| Name | BDBM50227020 |
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| Synonyms: | CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate |
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| Type | Small organic molecule |
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| Emp. Form. | C20H12ClN2O5S |
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| Mol. Mass. | 427.838 |
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| SMILES | Nc1c(cc(Nc2cccc(Cl)c2)c2C(=O)c3ccccc3C(=O)c12)S([O-])(=O)=O |
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| Structure | 
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