| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50347177 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_753740 (CHEMBL1799577) |
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| Ki | 0.2±n/a nM |
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| Citation |  Yamamoto, N; Fujii, H; Nemoto, T; Nakajima, R; Momen, S; Izumimoto, N; Hasebe, K; Mochizuki, H; Nagase, H Synthesis of new opioid derivatives with a propellane skeleton and their pharmacology: part 1. Bioorg Med Chem Lett21:4104-7 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50347177 |
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| n/a |
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| Name | BDBM50347177 |
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| Synonyms: | CHEMBL1797687 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H29NO2 |
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| Mol. Mass. | 315.4498 |
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| SMILES | CCC12CCN(CC3(O)CC3)[C@H](Cc3ccc(O)cc13)C2(C)C |r,THB:6:5:20:19.13.12| |
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| Structure | 
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