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TargetRelaxin-3 receptor 1
LigandBDBM50383001
Substrate/Competitorn/a
Meas. Tech.ChEMBL_818425 (CHEMBL2034745)
Ki>10000±n/a nM
Citation Shabanpoor, F; Akhter Hossain, M; Ryan, PJ; Belgi, A; Layfield, S; Kocan, M; Zhang, S; Samuel, CS; Gundlach, AL; Bathgate, RA; Separovic, F; Wade, JD Minimization of human relaxin-3 leading to high-affinity analogues with increased selectivity for relaxin-family peptide 3 receptor (RXFP3) over RXFP1. J Med Chem55:1671-81 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Relaxin-3 receptor 1
Name:Relaxin-3 receptor 1
Synonyms:G protein-coupled receptor SALPR | G-protein coupled receptor GPCR135 | GPCR135 | RL3R1_HUMAN | RLN3 receptor 1 | RLN3R1 | RXFP3 | Relaxin family peptide receptor 3 | SALPR | Somatostatin- and angiotensin-like peptide receptor
Type:PROTEIN
Mol. Mass.:51139.41
Organism:Homo sapiens (Human)
Description:ChEMBL_818423
Residue:469
Sequence:
MQMADAATIATMNKAAGGDKLAELFSLVPDLLEAANTSGNASLQLPDLWWELGLELPDGA
PPGHPPGSGGAESADTEARVRILISVVYWVVCALGLAGNLLVLYLMKSMQGWRKSSINLF
VTNLALTDFQFVLTLPFWAVENALDFKWPFGKAMCKIVSMVTSMNMYASVFFLTAMSVTR
YHSVASALKSHRTRGHGRGDCCGRSLGDSCCFSAKALCVWIWALAALASLPSAIFSTTVK
VMGEELCLVRFPDKLLGRDRQFWLGLYHSQKVLLGFVLPLGIIILCYLLLVRFIADRRAA
GTKGGAAVAGGRPTGASARRLSKVTKSVTIVVLSFFLCWLPNQALTTWSILIKFNAVPFS
QEYFLCQVYAFPVSVCLAHSNSCLNPVLYCLVRREFRKALKSLLWRIASPSITSMRPFTA
TTKPEHEDQGLQAPAPPHAAAEPDLLYYPPGVVVYSGGRYDLLPSSSAY
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  Blast E-value cutoff:
BDBM50383001
n/a
NameBDBM50383001
Synonyms:CHEMBL2030692
TypeSmall organic molecule
Emp. Form.C129H207N43O33S2
Mol. Mass.2952.422
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Structure
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