| Reaction Details |
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 | Report a problem with these data |
| Target | Relaxin-3 receptor 1 |
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| Ligand | BDBM50382992 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_818423 (CHEMBL2034650) |
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| IC50 | 5.13±n/a nM |
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| Citation |  Shabanpoor, F; Akhter Hossain, M; Ryan, PJ; Belgi, A; Layfield, S; Kocan, M; Zhang, S; Samuel, CS; Gundlach, AL; Bathgate, RA; Separovic, F; Wade, JD Minimization of human relaxin-3 leading to high-affinity analogues with increased selectivity for relaxin-family peptide 3 receptor (RXFP3) over RXFP1. J Med Chem55:1671-81 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Relaxin-3 receptor 1 |
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| Name: | Relaxin-3 receptor 1 |
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| Synonyms: | G protein-coupled receptor SALPR | G-protein coupled receptor GPCR135 | GPCR135 | RL3R1_HUMAN | RLN3 receptor 1 | RLN3R1 | RXFP3 | Relaxin family peptide receptor 3 | SALPR | Somatostatin- and angiotensin-like peptide receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 51139.41 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_818423 |
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| Residue: | 469 |
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| Sequence: | MQMADAATIATMNKAAGGDKLAELFSLVPDLLEAANTSGNASLQLPDLWWELGLELPDGA
PPGHPPGSGGAESADTEARVRILISVVYWVVCALGLAGNLLVLYLMKSMQGWRKSSINLF
VTNLALTDFQFVLTLPFWAVENALDFKWPFGKAMCKIVSMVTSMNMYASVFFLTAMSVTR
YHSVASALKSHRTRGHGRGDCCGRSLGDSCCFSAKALCVWIWALAALASLPSAIFSTTVK
VMGEELCLVRFPDKLLGRDRQFWLGLYHSQKVLLGFVLPLGIIILCYLLLVRFIADRRAA
GTKGGAAVAGGRPTGASARRLSKVTKSVTIVVLSFFLCWLPNQALTTWSILIKFNAVPFS
QEYFLCQVYAFPVSVCLAHSNSCLNPVLYCLVRREFRKALKSLLWRIASPSITSMRPFTA
TTKPEHEDQGLQAPAPPHAAAEPDLLYYPPGVVVYSGGRYDLLPSSSAY
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| BDBM50382992 |
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| n/a |
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| Name | BDBM50382992 |
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| Synonyms: | CHEMBL2030701 |
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| Type | Small organic molecule |
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| Emp. Form. | C166H262N50O46S4 |
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| Mol. Mass. | 3822.424 |
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| SMILES | n/a |
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| Structure | 
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