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TargetRegulator of G-protein signaling 8
LigandBDBM50384743
Substrate/Competitorn/a
Meas. Tech.ChEMBL_821036 (CHEMBL2039223)
IC50 7500±n/a nM
Citation Turner, EMBlazer, LLNeubig, RRHusbands, SM Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins. ACS Med Chem Lett3:146-150 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Regulator of G-protein signaling 8
Name:Regulator of G-protein signaling 8
Synonyms:RGS8 | RGS8_HUMAN | Regulator of G-protein signaling 8 (RGS8)
Type:Enzyme Catalytic Domain
Mol. Mass.:20925.80
Organism:Homo sapiens (Human)
Description:gi_74355113
Residue:180
Sequence:
MAALLMPRRNKGMRTRLGCLSHKSDSCSDFTAILPDKPNRALKRLSTEEATRWADSFDVL
LSHKYGVAAFRAFLKTEFSEENLEFWLACEEFKKTRSTAKLVSKAHRIFEEFVDVQAPRE
VNIDFQTREATRKNLQEPSLTCFDQAQGKVHSLMEKDSYPRFLRSKMYLDLLSQSQRRLS
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BDBM50384743
n/a
NameBDBM50384743
Synonyms:CHEMBL2037235
TypeSmall organic molecule
Emp. Form.C16H14N2O2S
Mol. Mass.298.36
SMILESCc1ccc(cc1)-n1sc(=O)n(Cc2ccccc2)c1=O
Structure
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