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TargetRegulator of G-protein signaling 4
LigandBDBM50384751
Substrate/Competitorn/a
Meas. Tech.ChEMBL_821035 (CHEMBL2039222)
IC50 7.2±n/a nM
Citation Turner, EMBlazer, LLNeubig, RRHusbands, SM Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins. ACS Med Chem Lett3:146-150 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4
Synonyms:RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM50384751
n/a
NameBDBM50384751
Synonyms:CHEMBL2037350
TypeSmall organic molecule
Emp. Form.C17H16N2O2S
Mol. Mass.312.386
SMILESCc1ccc(Cn2sc(=O)n(Cc3ccccc3)c2=O)cc1
Structure
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