| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 4 |
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| Ligand | BDBM50385164 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_822043 (CHEMBL2040206) |
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| Ki | 70±n/a nM |
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| Citation |  Baber, JC; Lowe, R; Saunders, J; Feher, M Automated generation of turn mimetics: proof of concept study for the MC4 receptor. Bioorg Med Chem20:3565-74 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 4 |
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| Name: | Melanocortin receptor 4 |
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| Synonyms: | MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36949.50 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32245 |
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| Residue: | 332 |
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| Sequence: | MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLL
ENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVN
IDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVS
GILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGAN
MKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPL
IYALRSQELRKTFKEIICCYPLGGLCDLSSRY
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| BDBM50385164 |
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| n/a |
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| Name | BDBM50385164 |
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| Synonyms: | CHEMBL2035944 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H34Cl2N4O2 |
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| Mol. Mass. | 529.501 |
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| SMILES | Clc1ccc(CNC(=O)[C@H]2CN(CC3CC3)C[C@H]2C(=O)NC2CCN(Cc3ccccc3)C2)c(Cl)c1 |r| |
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| Structure | 
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