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TargetDelta-type opioid receptor
LigandBDBM50391603
Substrate/Competitorn/a
Meas. Tech.ChEMBL_850392 (CHEMBL2150812)
Ki 0.151±n/a nM
Citation Ida, YMatsubara, ANemoto, TSaito, MHirayama, SFujii, HNagase, H Synthesis of quinolinomorphinan derivatives as highly selectived opioid receptor ligands. Bioorg Med Chem20:5810-31 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Delta-type opioid receptor
Name:Delta-type opioid receptor
Synonyms:DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:Enzyme Catalytic Domain
Mol. Mass.:40577.25
Organism:MOUSE
Description:P32300
Residue:372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50391603
n/a
NameBDBM50391603
Synonyms:CHEMBL2147916
TypeSmall organic molecule
Emp. Form.C25H26N2O3
Mol. Mass.402.4855
SMILESCOc1cccc2nc3C[C@]45CCN(C)[C@H](Cc6ccc(O)cc46)[C@]5(O)Cc3cc12 |r,TLB:14:13:24:23.17.16|
Structure
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